Copper-catalyzed intramolecular N-arylation of quinazolinones: Facile convergent approach to (-)-circumdatins H and J

Umesh A. Kshirsagar; Narshinha P. Argade

doi:10.1021/ol101597p

Copper-catalyzed intramolecular N-arylation of quinazolinones: Facile convergent approach to (-)-circumdatins H and J

Umesh A. Kshirsagar, Narshinha P. Argade

Research output: Contribution to journal › Article › peer-review

72 Scopus citations

Abstract

A copper-catalyzed intramolecular N-arylation of a quinazolinone nucleus that furnished the central benzodiazepine core unit has been demonstrated to accomplish an efficient convergent total synthesis of (-)-circumdatins H and J.

Original language	English
Pages (from-to)	3716-3719
Number of pages	4
Journal	Organic Letters
Volume	12
Issue number	16
DOIs	https://doi.org/10.1021/ol101597p
State	Published - 20 Aug 2010
Externally published	Yes

ASJC Scopus subject areas

Biochemistry
Physical and Theoretical Chemistry
Organic Chemistry

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10.1021/ol101597p

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title = "Copper-catalyzed intramolecular N-arylation of quinazolinones: Facile convergent approach to (-)-circumdatins H and J",

abstract = "A copper-catalyzed intramolecular N-arylation of a quinazolinone nucleus that furnished the central benzodiazepine core unit has been demonstrated to accomplish an efficient convergent total synthesis of (-)-circumdatins H and J.",

author = "Kshirsagar, {Umesh A.} and Argade, {Narshinha P.}",

year = "2010",

month = aug,

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doi = "10.1021/ol101597p",

language = "English",

volume = "12",

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journal = "Organic Letters",

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T2 - Facile convergent approach to (-)-circumdatins H and J

AU - Kshirsagar, Umesh A.

AU - Argade, Narshinha P.

PY - 2010/8/20

Y1 - 2010/8/20

N2 - A copper-catalyzed intramolecular N-arylation of a quinazolinone nucleus that furnished the central benzodiazepine core unit has been demonstrated to accomplish an efficient convergent total synthesis of (-)-circumdatins H and J.

AB - A copper-catalyzed intramolecular N-arylation of a quinazolinone nucleus that furnished the central benzodiazepine core unit has been demonstrated to accomplish an efficient convergent total synthesis of (-)-circumdatins H and J.

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U2 - 10.1021/ol101597p

DO - 10.1021/ol101597p

M3 - Article

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AN - SCOPUS:77955677822

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VL - 12

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JO - Organic Letters

JF - Organic Letters

IS - 16

ER -

Copper-catalyzed intramolecular N-arylation of quinazolinones: Facile convergent approach to (-)-circumdatins H and J

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