Cyclic endiamino peptides: A new synthesis of imidazopyrazines

Yael Kogon; Lee Goren; Doron Pappo; Amira Rudi; Yoel Kashman

doi:10.1002/ejoc.200900008

Cyclic endiamino peptides: A new synthesis of imidazopyrazines

Yael Kogon, Lee Goren, Doron Pappo, Amira Rudi, Yoel Kashman

Research output: Contribution to journal › Article › peer-review

5 Scopus citations

Abstract

By applying the cyclic endiamino cyclisation methodology to linear tripeptides embodying a β-turn-directing amino acid, the imidazopyrazine ring system was afforded. A mechanism involving the originally desired nine-membered cyclic encliamine is suggested.

Original language	English
Pages (from-to)	1852-1854
Number of pages	3
Journal	European Journal of Organic Chemistry
Issue number	12
DOIs	https://doi.org/10.1002/ejoc.200900008
State	Published - 1 Apr 2009
Externally published	Yes

Keywords

Cyclization
Enols
Nitrogen heterocycles
Peptides

ASJC Scopus subject areas

Physical and Theoretical Chemistry
Organic Chemistry

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10.1002/ejoc.200900008

Cite this

@article{56727d54592b4ea7bcc927ed30681e41,

title = "Cyclic endiamino peptides: A new synthesis of imidazopyrazines",

abstract = "By applying the cyclic endiamino cyclisation methodology to linear tripeptides embodying a β-turn-directing amino acid, the imidazopyrazine ring system was afforded. A mechanism involving the originally desired nine-membered cyclic encliamine is suggested.",

keywords = "Cyclization, Enols, Nitrogen heterocycles, Peptides",

author = "Yael Kogon and Lee Goren and Doron Pappo and Amira Rudi and Yoel Kashman",

year = "2009",

month = apr,

day = "1",

doi = "10.1002/ejoc.200900008",

language = "English",

pages = "1852--1854",

journal = "European Journal of Organic Chemistry",

issn = "1434-193X",

publisher = "John Wiley and Sons Ltd",

number = "12",

}

TY - JOUR

T1 - Cyclic endiamino peptides

T2 - A new synthesis of imidazopyrazines

AU - Kogon, Yael

AU - Goren, Lee

AU - Pappo, Doron

AU - Rudi, Amira

AU - Kashman, Yoel

PY - 2009/4/1

Y1 - 2009/4/1

N2 - By applying the cyclic endiamino cyclisation methodology to linear tripeptides embodying a β-turn-directing amino acid, the imidazopyrazine ring system was afforded. A mechanism involving the originally desired nine-membered cyclic encliamine is suggested.

AB - By applying the cyclic endiamino cyclisation methodology to linear tripeptides embodying a β-turn-directing amino acid, the imidazopyrazine ring system was afforded. A mechanism involving the originally desired nine-membered cyclic encliamine is suggested.

KW - Cyclization

KW - Enols

KW - Nitrogen heterocycles

KW - Peptides

UR - http://www.scopus.com/inward/record.url?scp=63849286281&partnerID=8YFLogxK

U2 - 10.1002/ejoc.200900008

DO - 10.1002/ejoc.200900008

M3 - Article

AN - SCOPUS:63849286281

SN - 1434-193X

SP - 1852

EP - 1854

JO - European Journal of Organic Chemistry

JF - European Journal of Organic Chemistry

IS - 12

ER -

Cyclic endiamino peptides: A new synthesis of imidazopyrazines

Abstract

Keywords

ASJC Scopus subject areas

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